program | The 27th French-Japanese Symposium on Medicinal and Fine Chemistry

FJS2019 in Fukuoka Program

The program is composed of invited lectures, a poster session and related discussions. All lectures are by invitation. The symposium language will be English. Plenary lectures will last 50 min (40+10), invited lectures will last 30 min (25+5).

Sunday, May 19, 2019
15:00	Registration at Hotel Leopalace Posting the Posters
17:30	L1 Hirosato Kondo (National Institute of Biomedical Innovation, Health and Nutrition) Current Topics & Future Direction of Drug Discovery Research http://www.nibiohn.go.jp/en/cddr/about/	Chair: Shigeki Sasaki
19:00	Welcome Mixer at Hotel Leopalace
Monday, May 20, 2019
8:30	Opening Remarks: Shigeki Sasaki
8:40	L2 Alain WAGNER (Université de Strasbourg) Interfacing living and synthetic systems at the molecular level www.biofunctional.eu	Chair:
9:30	S1 Masanao INAGAKI (Shionogi) Discovery of naldemedine: A potent and orally available opioid receptor antagonist for treatment of opioid-induced adverse effects	Chair:
10:00	Coffee Break
10:30	L3 Sylviane SABO-ETIENNE (LCC CNRS Toulouse) Dihydrogen and Polyfunctional Ligands: Tools for Applications in Catalysis https://www.lcc-toulouse.fr/article474.html	Chair:
11:20	S2 Daisuke TANAKA(Exscientia Ltd) Re-energising Small Molecule Drug Discovery by Centaur Chemist™
11:50	Lunch
13:20	L4 Takayoshi SUZUKI (Kyoto Prefectural University of Medicine) Chemical Control of Epigenetics for the Treatment of Cancers and Neurological Disorders http://www.f.kpu-m.ac.jp/y/chemistry/English/suzuki.html	Chair:
14:10	S3 Sébastien LEMAIRE (Janssen Pharmaceutical Companies of Johnson & Johnson) Stereoselective C-Glycosylation Reactions with Arylzinc Reagents, Application to Canagliflozin Synthesis and Mechanistic Study	Chair:
14:40	Coffee Break
15:10	L5 Masaya SAWAMURA (Hokkaido University) Ligand-Enabled Selective Borylation of C(sp2)–H and C(sp3)–H Bond http://wwwchem.sci.hokudai.ac.jp/~orgmet/index.php?id=25	Chair:
16:00	S4 Christophe Morice (Prestwick Chemical) Foliglurax, a novel mGluR4 positive allosteric modulator: Successful medicinal chemistry strategy from hit to candidate	Chair:
16:30	Poster Session with Oral Presentation
19:00	Refreshment in the Hakata Down Town
Tuesday, May 21, 2019
8:30	L6 Takeshi WADA (Tokyo University of Science) Stereocontrolled synthesis and properties of phosphorus modified nucleic acid drugs https://www.tus.ac.jp/en/fac/p/index.php?6791	Chair:
9:20	S5 Guillaume BERTHON (Syngenta) Where do new agrochemicals come from?
9:50	Coffee Break
10:20	S6 Taro TERAUCHI (Eisai) Discovery of a novel and potent dual orexin 1/orexin 2 receptor antagonist, Lemborexant (E2006), for the treatment of sleep disorders
10:50	S7 Jidong ZHANG (Sanofi) Sequanamycin, a new class of potent oral active anti-tuberculosis Macrolides	Chair:
11:20	S8 Tohru KAMBE (Ono) Discovery of Potent, Selective Prostaglandin FP/EP3 Dual Agonist, DE-126/ONO-9054, for the Treatment of Glaucoma	Chair:
11:50	Lunch
13:20	L7 Chantal ANDRAUD (ENS Lyon) To be announced http://www.ens-lyon.fr/CHIMIE/laboratory/directory/andraud-chantal	Chair:
14:10	S9 Thierry BILLARD (University Claude Bernard - Lyon 1) From radiochemistry to medical imaging: a travel in PET imaging world http://fmi-lyon.bcpmdb.com	Chair:
14:40	Move to Touchouji-Temple
	Touchou-ji Temple The oldest temple in Japan that Kukai (Kobo Daishi) built in the year of 806. A large wooden Buddha over 10 meters. The tombs of Kuroda family who governed Fukuoka area during Edo Age (17-19 century). https://yokanavi.com/en/spot/26928/
	Bus or walk to Hakata Bay-side
16:25	Twilight Cruise (1 hr 30) https://www.mariera.jp/fl/en/
19:00	Banquet Hakata Hyakunengura (Ishikura Sake Brewery) https://yokanavi.com/en/spot/26972/
Wednesday, May 22, 2019
8:30	L8 Hiroki OGURI (Tokyo Univ. of Agriculture and Technology) Artificial assembly lines for divergent syntheses of natural products and their variants http://web.tuat.ac.jp/~h_oguri/en/index.html	Chair:
9:20	S10 Tatiana BESSET (INSA de Rouen, Université de Rouen) Recent advances to access fluorinated scaffolds http://sciences-techniques.univ-rouen.fr/tatiana-besset-530552.kjsp	Chair:
9:50	Coffee Break
10:20	L9 Michael SMIETANA (IBMM Montpellier) DNA as a Versatile Chemical Scaffold for Recognition, Assembly and Asymmetric Catalysis https://sites.google.com/site/michaelsmietanaum2/	Chair:
11:10	S11 Takahiko TANIGUCHI (Takeda) Discovery of Clinical Candidate TAK-915, A Highly Potent, Selective, and Brain-Penetrating Phosphodiesterase 2A Inhibitor for the Treatment of Cognitive Disorders	Chair:
11:40	Closing
12:30	Departure to Post-Symposium Tour